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Indoles from simple anilines and alkynes: palladium-catalyzed C-H activation using dioxygen as the oxidant.
Angew Chem Int Ed Engl. 2009; 48(25):4572-6.AC

Abstract

Pd doles it out: A palladium-catalyzed approach to indoles using the title reaction was achieved (see scheme). The oxidant used in this catalytic cycle was O(2). Both N-nonsubstituted and N-alkyl monosubstituted anilines can be successfully transformed into the corresponding indoles by this method.

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Publisher Full Text (DOI)

Authors+Show Affiliations

Shi Z
State Key Laboratory of Natural and Biomimetic Drugs, Peking University, School of Pharmaceutical Sciences, Peking University, Xue Yuan Rd. 38, Beijing 100083, China.
Zhang C
No affiliation info available
Li S
No affiliation info available
Pan D
No affiliation info available
Ding S
No affiliation info available
Cui Y
No affiliation info available
Jiao N
No affiliation info available

MeSH

AlkynesAniline CompoundsCatalysisCyclizationIndolesOxidantsOxygenPalladium

Pub Type(s)

Journal Article
Research Support, Non-U.S. Gov't

Language

eng

PubMed ID

19444850

Citation

Shi, Zhuangzhi, et al. "Indoles From Simple Anilines and Alkynes: Palladium-catalyzed C-H Activation Using Dioxygen as the Oxidant." Angewandte Chemie (International Ed. in English), vol. 48, no. 25, 2009, pp. 4572-6.
Shi Z, Zhang C, Li S, et al. Indoles from simple anilines and alkynes: palladium-catalyzed C-H activation using dioxygen as the oxidant. Angew Chem Int Ed Engl. 2009;48(25):4572-6.
Shi, Z., Zhang, C., Li, S., Pan, D., Ding, S., Cui, Y., & Jiao, N. (2009). Indoles from simple anilines and alkynes: palladium-catalyzed C-H activation using dioxygen as the oxidant. Angewandte Chemie (International Ed. in English), 48(25), 4572-6. https://doi.org/10.1002/anie.200901484
Shi Z, et al. Indoles From Simple Anilines and Alkynes: Palladium-catalyzed C-H Activation Using Dioxygen as the Oxidant. Angew Chem Int Ed Engl. 2009;48(25):4572-6. PubMed PMID: 19444850.
* Article titles in AMA citation format should be in sentence-case
TY - JOUR T1 - Indoles from simple anilines and alkynes: palladium-catalyzed C-H activation using dioxygen as the oxidant. AU - Shi,Zhuangzhi, AU - Zhang,Chun, AU - Li,Si, AU - Pan,Delin, AU - Ding,Shengtao, AU - Cui,Yuxin, AU - Jiao,Ning, PY - 2009/5/16/entrez PY - 2009/5/16/pubmed PY - 2009/7/31/medline SP - 4572 EP - 6 JF - Angewandte Chemie (International ed. in English) JO - Angew Chem Int Ed Engl VL - 48 IS - 25 N2 - Pd doles it out: A palladium-catalyzed approach to indoles using the title reaction was achieved (see scheme). The oxidant used in this catalytic cycle was O(2). Both N-nonsubstituted and N-alkyl monosubstituted anilines can be successfully transformed into the corresponding indoles by this method. SN - 1521-3773 UR - https://www.unboundmedicine.com/medline/citation/19444850/Indoles_from_simple_anilines_and_alkynes:_palladium_catalyzed_C_H_activation_using_dioxygen_as_the_oxidant_ L2 - https://doi.org/10.1002/anie.200901484 DB - PRIME DP - Unbound Medicine ER -